Almitrine dimesylate
CAS No. 29608-49-9
Almitrine dimesylate ( Almitrine mesylate;Almitrine bismesylate;Almitrine bismethanesulfonate )
产品货号. M20572 CAS No. 29608-49-9
Almitrine dimesylate inhibits selectively the Ca2+-dependent K+ channel and that in rat chemoreceptor cellsused in the treatment of hypoxemic chronic lung diseases.
纯度: >98% (HPLC)
规格 | 价格/人民币 | 库存 | 数量 |
25MG | ¥284 | 有现货 |
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50MG | ¥373 | 有现货 |
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100MG | ¥632 | 有现货 |
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200MG | ¥875 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Almitrine dimesylate
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Almitrine dimesylate inhibits selectively the Ca2+-dependent K+ channel and that in rat chemoreceptor cellsused in the treatment of hypoxemic chronic lung diseases.
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产品描述Almitrine dimesylate inhibits selectively the Ca2+-dependent K+ channel and that in rat chemoreceptor cellsused in the treatment of hypoxemic chronic lung diseases.
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同义词Almitrine mesylate;Almitrine bismesylate;Almitrine bismethanesulfonate
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通路Cell Cycle/DNA Damage
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靶点Potassium Channel
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受体Potassium Channel
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研究领域Metabolic Disease
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适应症chronic obstructive pulmonary disease
化学信息
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CAS Number29608-49-9
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分子量669.76
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分子式C28H37F2N7O6S2
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纯度>98% (HPLC)
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溶解度DMSO:125 mg/mL (186.63 mM)
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SMILESCS(O)(=O)=O.CS(O)(=O)=O.Fc1ccc(cc1)C(N1CCN(CC1)c1nc(NCC=C)nc(NCC=C)n1)c1ccc(F)cc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
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TKIM
TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.TKIM binds to the pocket of the IM state of TREK-1, which differs from the binding of common inhibitors, which bind to channels in the inactive state.?
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Pinacidil monohydrat...
Pinacidil monohydrate is a potassium channel activator, antihypertensive drug.Pinacidil hydrate activates the ATP-modulated potassium channels of guinea pog bladder and heart with Ki of 104 and 251 nM, respectively.
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Glibornuride
Glibornuride is a blocker of ATP-sensitive K+ channel(pKi: 5.75). Glibornuride inhibits high affinity [3H]-glibenclamide binding with the potencies expected from their K+ channel activity.